Partenaires

Logo Chimiothèque Nationale
CNRS

Plaquette de la CN

plaquette


Rechercher

Sur ce site


Sur le Web du CNRS




Certification ISO 9001:2008

iso


Accueil du site > Publications > 2- Criblages de chimiothèques > 2016

Publications 2016

1. Grandin, C., Hourani, M. L., Janin, Y. L., Dauzonne, D., Munier-Lehmann, H., Paturet, A., Taborik, F., Vabret, A., Contamin, H., Tangy, F. and Vidalain, P. O.
Respiratory syncytial virus infection in macaques is not suppressed by intranasal sprays of pyrimidine biosynthesis inhibitors
Antiviral Research 2016, 125, 58-62.

2. Petrella, S., Aubry, A., Janvier, G., Coutant, E. P., Cartier, A., Dao, T.-H., Bonhomme, F. J., Motreff, L., Pissis, C., Bizet, C., Clermont, D., Begaud, E., Retailleau, P., Munier-Lehmann, H., Capton, E., Mayer, C. and Janin, Y. L.
Synthesis and evaluation of original bioisosteres of bacterial type IIA topoisomerases inhibitors
Canadian Journal of Chemistry 2016, 94, 240-250.

3. Raj, S. ; Krishnan, K. ; Askew, D. S. ; Helynck, O. ; Suzanne, P. ; Lesnard, A. ; Rault, S. ; Zeidler, U. ; D’Enfert, C. ; Latgé, J.-P. ; Munier-Lehmann, H. ; Saveanu, C.
The Toxicity of a Novel Antifungal Compound Is Modulated by Endoplasmic Reticulum- Associated Protein Degradation Components
Antimicrob. Agents Chemother. 2016, 60, 1438–1449.

4. Gellis, A. ; Primas, N. ; Hutter, S. ; Lanzada, G. ; Remusat, V. ; Verhaeghe, P., P. ; Vanelle, P. ; Azas, N.
Looking for new antiplasmodial quinazolines : DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum
Eur. J. Med. Chem. 2016, 119, 34-44.

5. Da Costa, L. ; Roche, M. ; Scheers, E. ; Coluccia, A. ; Neyts, J. ; Terme, T. ; Leyssen, P. ; Silvestri, R. ; Vanelle, Patrice
VP1 crystal structure-guided exploration and optimization of 4,5-dimethoxybenzene-based inhibitors of rhinovirus 14 infection
Eur. J. Med. Chem. 2016, 115, 453-462.

6. R. Quillet, S. Ayachi, F. Bihel, K. Elhabazi, B. Ilien, F. Simonin
RF-Amide Neuropeptides And Their Receptors In Mammals : Pharmacological Properties, Drug Development And Main Physiological Functions
Pharmacol. Ther., 2016, 160, 84-132.

7. I. Buffel, A. Meurs, J. Portelli, R. Raedt, V. De Herdt, L. Poppe, V. De Meulenaere, W. Wadman, F. Bihel, M. Schmitt, K. Vonck, J.J. Bourguignon, F. Simonin, I. Smolders and P. Boon
The effect of neuropeptide FF in the amygdala kindling model
Eur. J. Med. Acta Neurologica Scandinavica 2016, 134(3):181-8.

8. Vehary Sakanyan, Philippe Hulin, Rodolphe Alves de Sousa, Viviane A. O. Silva, Artur Hambardzumyan, Steven Nedellec, Christophe Tomasoni, Cédric Logé, Charles Pineau, Christos Roussakis, Fabrice Fleury & Isabelle Artaud
Activation of EGFR by small compounds through coupling the generation of hydrogen peroxide to stable dimerization of Cu/Zn SOD1
Scientific Reports 2016, doi:10.1038/srep21088.

9. L. Saint-Paul, C.-H. Nguyen, A. Buffière, J.-P. P. d. Barros, A. Hammann, C. Landras-Guetta, R. Filomenko, M.-L. Chrétien, P. Johnson, J.-N. Bastie, L. Delva and R. Quéré
CD45 phosphatase is crucial for human and murine acute myeloid leukemia maintenance through its localization in lipid rafts
Oncotarget, 2016, 7.

10. Labriere, C. ; Talapatra, S. K., Thoret, S., Bougeret, C., Kozielski, F., Guillou, C.
New MKLP-2 Inhibitors in the Paprotrain Series : Design, Synthesis and Biological Evaluation
Bioorg. Med. Chem. 2016, 24, 721-734.
DOI : 10.1016/j.bmc.2015.12.042.

Mise à jour le 10 janvier 2017