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Accueil du site > Publications > 2- Criblages de chimiothèques > 2014

Publications 2014

1. A. Caruso, M.S. Sinicropi, J.-C. Lancelot, H. El-Kashef, C. Saturnino, G. Aubert, C. Ballandonne, A. Lesnard, T. Cresteil, P. Dallemagne, S. Rault
Synthesis end Evaluation of cytotoxic activities of novel guanidines derived from carbazoles
Bioorganic and Medicinal Chemistry Letters, 2014, 24, 467 - 472.

2. F. Fontaine, A. Hequet, A.-S. Voisin-Chiret, A. Bouillon, A. Lesnard, T. Cresteil, C. Jolivalt, S. Rault
First identification of heterocyclic boronic acids as novel potential inhibitors of the Staphylococcus aureus NorA efflux pump
Journal of Medicinal Chemistry, 2014, 57, (6), 2536-2548.

3. N. Primas, P. Suzanne, P. Verhaeghe, S. Hutter, C. Kieffer, M. Laget, A. Cohen, J. Broggi, J.-C. Lancelot, A. Lesnard, P. Dallemagne, P. Rathelot, S. Rault, P. Vanelle, N. Azas
Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents
European Journal of Medicinal Chemistry, 2014, 83, 26-35.

4. J. F. Margathe, X. Iturrioz, R. Alvear-Perez, C. Marsol, S. Riche, H. Chabane, N. Tounsi, M. Kuhry, D. Heissler, M. Hibert, C. Llorens-Cortes, D. Bonnet
Structure Activity Relationship Studies toward the Discovery of Selective Apelin Receptor Agonists
J Med Chem, 2014, 57, 2908-2919.

5. D. Horvath, M. Lisurek, B. Rupp, R. Kuhne, E. Specker, J. von Kries, D. Rognan, C. D. Andersson, F. Almqvist, M. Elofsson, P. A. Enqvist, A. L. Gustavsson, N. Remez, J. Mestres, G. Marcou, A. Varnek, M. Hibert, J. Quintana, R. Frank
Design of a General-Purpose European Compound Screening Library for EU-OPENSCREEN
ChemMedChem, 2014, 9, 2309-2326.

6. Vehary Sakanyan, Marie Angelini, Mickael Le Béchec, Michèle Françoise Lecocq, Florence Benaiteau, Bénédicte Rousseau, Aram Gyulkhandanyan, Lusine Gyulkhandanyan, Cédric Logé, Eric Reiter, Christos Roussakis & Fabrice Fleury
Screening and discovery of nitro-benzoxadiazole compounds activating epidermal growth factor receptor (EGFR) in cancer cells
Scientific Reports 4, 2014, doi:10.1038/srep03977.

7. Montana, M. ; Correard, F. ; Khoumeri, O. ; Esteve, M.-A. ; Terme, T. ; Vanelle, P.
Synthesis of new quinoxalines containing an oxirane ring by the TDAE strategy and in vitro evaluation in neuroblastoma cell lines
Molecules 2014, 19, 14987-14998.

8. Tabele, C. ; Cohen, A. ; Curti, C. ; Bouhlel, A. ; Hutter, S. ; Remusat, V. ; Primas, N. ; Terme, T. ; Azas, N. ; Vanelle, P.
New series of monoamidoxime derivatives displaying versatile antiparasitic activity
European Journal of Medicinal Chemistry 2014, 87, 440-453.

9. Crozet, M. ; D. ; Terme, T. ; Vanelle, P.
Designing New 5-Nitroimidazoles : Towards Safer Anti-infectious Agents
Letters in Drug Design & Discovery 2014, 11, 531-559..

10. Roche, M. ; Lacroix, C. ; Khoumeri, O. ; Franco, D. ; Neyts, J. ; Terme, T. ; Leyssen, P. ; Vanelle, P.
Synthesis, biological activity and structure-activity relationship of 4,5-dimethoxybenzene derivatives inhibitor of rhinovirus 14 infection
European Journal of Medicinal Chemistry 2014, 76, 445-459..

Mise à jour le 10 janvier 2017