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Accueil du site > Publications > 2- Criblages de chimiothèques > 2013

Publications 2013

1. Ada Collura, Laetitia Marisa, Diletta Trojan, Olivier Buhard, Anaïs Lagrange, Arnaud Saget, Marianne Bombled, Patricia Méchighel, Mira Ayadi, Martine Muleris, Aurélien de Reynies, Magali Svrcek, Jean-Francois Fléjou, Jean-Claude Florent, Florence Mahuteau-Betzer, Anne-Marie Faussat, Alex Duval
Extensive characterization of sphere models established from colorectal cancer cell lines
Cell. Mol. Life Sci. 2013,117 (2), 316-323.

2. Le Ly, TT., Vu, H.L., Naud-Martin, D., Bombled, M., Nguyen, C.H., and Molla A.
New hydrosoluble benzo[e]pyridoindolones as potent inhibitors of aurora kinases
Chem. Med. Chem. 2013, 8, 289-296.

3. Prudent, R., Vassal-Stermann, E., Nguyen, C.H., Mollaret, M., Viallet, J., Castan, A., Barette, C., Pillet, C., Martinez, A., Soleilhac, E., Feige, J-J., Billaud, M., Florent J-C., and Lafanechère, L.
Azaindole derivatives are inhibitors of microtubule dynamics, with anticancer and anti-angiogenic activities
Br J Pharmacol. 2013, 168, 673-685.

4. Lucas-Hourani M, Dauzonne D, Jorda P, Cousin G, Lupan A, Helynck O, Caignard G, Janvier G, André-Leroux G, Khiar S, Escriou N, Desprès P, Jacob Y, Munier-Lehmann H, Tangy F, Vidalain PO
Inhibition of pyrimidine biosynthesis pathway suppresses viral growth through innate immunity
PLoS Pathog. 2013 ;9(10):e1003678.

5. Ceccaldi A., Rajavelu A., Ragozin S., Sénamaud-Beaufort C., Bashtrykov P., Testa N., Dali-Ali H., Maulay-Bailly C., Amand S., Guianvarc’h D., Jeltsch A., Arimondo P.B.
Identification of novel inhibitors of DNA methylation by screening of a chemical library
ACS Chem Biol., 2013, 8(3), 543-8.

6. Since, Marc ; Freret, Thomas ; Nee, Gerald ; Terme, Thierry ; Vanelle, Patrice ; Boulouard, Michel
New orally effective 3-(2-nitro)phenylpropanamide analgesic derivatives : synthesis and antinociceptive evaluation
European Journal of Medicinal Chemistry, 2013, 69, 728-734.

7. Cohen, Anita ; Crozet, Maxime D. ; Rathelot, Pascal ; Azas, Nadine ; Vanelle, Patrice
Synthesis and promising in vitro antiproliferative activity of sulfones of a 5-nitrothiazole series
Molecules, 2013, 18, 97-113.

8. F. Daubeuf, M. Hachet-Haas, P. Gizzi, V. Gasparik, D. Bonnet, V. Utard, M. Hibert, N. Frossard, J. L. Galzi
An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice
J Biol Chem, 2013, 288, 11865-11876.

9. E. Audran, R. Dagher, S. Gioria, P. O. Tsvetkov, A. A. Kulikova, B. Didier, P. Villa A. A. Makarov M. C. Kilhoffer, J. Haiech
A general framework to characterize inhibitors of calmodulin : Use of calmodulin inhibitors to study the interaction between calmodulin and its calmodulin binding domains
BBA-Mol Cell Res, 2013, 1833, 1720-1731.

10. Munier-Lehmann, H., Vidalain, P. O., Tangy, F. and Janin, Y. L.
On dihydroorotate dehydrogenases and their inhibitors and uses
J. Med. Chem. 56, 3148-3167.

11. Raoul des Essarts, Y. ; Sabbah, M. ; Comte, A. ; Soulère, L. ; Queneau, Y. ; Hélias, V. ; Faure, F.
N,N’-alkylatedImidazolium- Derivatives act as Quorum-Sensing Inhibitors Targeting the Pectobacteriumatrosepticum-induced Symptoms on Potato Tubers
Int. J. Mol. Sci. 2013, 14, 19976-19986.

12. Since, Marc ; Freret, Thomas ; Nee, Gerald ; Terme, Thierry ; Vanelle, Patrice ; Boulouard, Michel
New orally effective 3-(2-nitro)phenylpropanamide analgesic derivatives : synthesis and antinociceptive evaluation
European Journal of Medicinal Chemistry 2013, 69, 728-734.

13. Cohen, Anita ; Crozet, Maxime D. ; Rathelot, Pascal ; Azas, Nadine ; Vanelle, Patrice
Synthesis and promising in vitro antiproliferative activity of sulfones of a 5-nitrothiazole series
Molecules 2013, 18, 97-113.

14. Magellana, H. ; Boccarab, M. ; Drujona, T. ; Souliéc, M.C. ; Guillou, C. ; Joëlle Dubois, J. ; Becker, H.F.
Discovery of two new inhibitors of Botrytis cinerea chitin synthase by a chemical library screening targeting the non-structural protein nsP2
Bioorg. Med. Chem. 2013, 21, 4997-5003.

15. Lucas-Hourani, M. ; Lupan, A. ; Desprès, P. ; Thoret, S. ; Pamlard, O. ; Dubois, J. ; Guillou, C. ;Tangy, F. ; Munier-Lehmann, H. ; Vidalain, P.O.
A phenotypic assay to identify chikungunya virus inhibitors
J. Biomol. Screen 2013, 18, 172-179.

16. Beury-Cirou, A. ; Tannières, M. ; Vandeputte, O. ; Minard, C. ; Soulère, L. ; Rasamiravaka, T. ; Dodd, R.H., Queneau, Y. ; Dessaux, Y. ; Guillou, C. ; Faure, D.
At a Supra-Physiological Concentration, Human Sexual Hormones Act as Quorum-Sensing Inhibitors
Plosone 2013, 8, 0083564 DOI : 10.1371.

Mise à jour le 10 janvier 2017