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Accueil du site > Publications > 2- Criblages de chimiothèques > 2010

Publications 2010

1. Prudent, R. ; Moucadel, V. ; Nguyen, C.H ; Barette, C. ; Schmidt, F. ; Florent, J.-C. ; Lafanechere, L. ; Sautel, C. F. ; Duchemin-Pelletier, E. ; Spreux, E. ; Filhol, O. ; Reiser, J.-B. ; Cochet, C.
Antitumor activity of pyridocarbazole and benzopyridoindole derivatives that inhibit protein kinase CK2
Cancer Research 2010, 70 (23), 9865-9874.

Targeting the cell cycle and the PI3K pathway : A possible universal strategy to reactivate innate tumor suppressor programmes in cancer cells
International Journal of Oncology 2010, 36, 873-881.

3. López-Ramos M, Prudent R, Moucadel V, Sautel CF, Barette C, Lafanechère L, Mouawad L, Grierson D, Schmidt F, Florent JC, Filippakopoulos P, Bullock AN, Knapp S, Reiser JB and Cochet C
New potent dual inhibitors of CK2 and Pim kinases : Discovery and structural insights
FASEB Journal 2010, 24 (9), 3171-3185.

4. Bouhlel, Ahlem ; Curti, Christophe ; Dumetre, Aurelien ; Laget, Michele ; Crozet, Maxime D. ; Azas, Nadine ; Vanelle, Patrice
Synthesis and evaluation of original amidoximes as antileishmanial agents _ Bioorganic & Medicinal Chemistry 2010, 18(20), 7310-7320.

5. Nadji-Boukrouche, Aida R. ; Khoumeri, Omar ; Terme, Thierry ; Liacha, Messaoud ; Vanelle, Patrice
Original TDAE reactivity in benzoxa- and benzothiazolone series
ARKIVOC (Gainesville, FL, United States) 2010,10, 358-370.

6. Maillard-Boyer, Martine ; Castera-Ducros, Caroline ; Verhaeghe, Pierre ; Sifredi, France ; Rathelot, Pascal ; Vanelle, Patrice
Access to original vinylic chlorides in the quinazoline series via a monoelectronic transfer reaction approach
Molecules 2010, 15, 2719-2729.

7. Juspin, Thierry ; Giuglio-Tonolo, Gamal ; Terme, Thierry ; Vanelle, Patrice
First TDAE-mediated double addition of nitrobenzylic anions to aromatic dialdehydes
Synthesis 2010, 5, 844-848.

8. Juspin, Thierry ; Laget, Michele ; Terme, Thierry ; Azas, Nadine ; Vanelle, Patrice TDAE-assisted synthesis of new imidazo[2,1-b]thiazole derivatives as anti-infectious agents European Journal of Medicinal Chemistry 2010, 45(2), 840-845.

9. Kabri, Youssef ; Azas, Nadine ; Dumetre, Aurelien ; Hutter, Sebastien ; Laget, Michele ; Verhaeghe, Pierre ; Gellis, Armand ; Vanelle, Patrice
Original quinazoline derivatives displaying antiplasmodial properties
European Journal of Medicinal Chemistry 2010, 45(2), 616-622.

10. V. Perri, C. Rochais, J. Sopkova-de Oliveira Santos, R. Legay, T. Cresteil, P. Dallemagne, S. Rault
Hydrogenative desulphurization of thienopyrrolizinones : An easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity
European Journal of Medicinal Chemistry, 2010, 45, 1146-1150.

11. J. Sopkova-de Oliveira Santos, A. Lesnard, J.-H. Agondanou, N. Dupont, A.-M. Godard, S. Stiebing, C. Rochais, F. Fabis, P. Dallemagne, R. Bureau, S. Rault
Virtual screening discovery of new acetylcholinesterase inhibitors issued from CERMN chemical library
Journal of Chemical Information and Modeling, 2010, 50(3), 422-428.

12. A. Lepailleur, S. Lemaitre, F. Xiao, J. Sopkova-de Oliveira Santos, P. Delagrange, J. Boutin, P. Renard, R. Bureau, S. Rault
Receptor- and ligand-based study on novel 2,2’-bithienyl derivatives as non-peptidic AANAT inhibitors
Journal of Chemical Information and Modeling, 2010, 50(3), 446-460.

13. D. Brossard, L. El Kihel, M. Clement, W. Sebbahi, M. Khalid, C. Roussakis, S. Rault
Synthesis of bile acid derivatives and in vitro cytotoxic activity with pro-apoptotic process on multiple myeloma (KMS-11), glioblastoma multiform (GBM), and colonic carcinoma (HCT-116) human cell lines
European Journal of Medicinal Chemistry, 2010, 45(7), 2912-2918.

14. T. Varin, H. Gutiérrez-de-Terán, M. Castro, J. Brea, F. Fabis, F. Dauphin, J. Aqvist, A. Lepailleur, P. Perez, J. Burgueño, J. Vela, M. Loza, J. Rodrigo
Phe369(7.38) at Human 5-HT7 Receptors Confers Interspecies Selectivity to Antagonists and Partial Agonists
British Journal of Pharmacology, 2010, 159, 1069-1081.

15. E. Laine, C. Goncalves, J. Karst, A. Lesnard, S. Rault, W.-J. Tang, T. E. Malliavin, D. Ladant, A. Blondel
The allostery as a target to find inhibitors of the calmodulin-induced activation of the Edema Factor from Bacillus anthracis
Proceedings of the National Academic Sciences, 2010, 107, (25), 11277-11282.

16. G. Pavé, S. Lazar, A. Lesnard, S. Rault, G. Guillaumet
Synthesis of aminopyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives as serotoninergic 5-HT7 ligands
Arkivoc, 2010, 10, 116-131.

17. Cailly T., Dumas N., Millet P., Lemaitre S., Fabis F., Charnay Y., Rault S
Synthesis and characterization of a iodine-125-labeled pyrrolo[1,2-a]thieno[3,2-e]pyrazine and evaluation as a potential 5-HT4R SPECT tracer
European Journal of Medicinal Chemistry (2010), 45(11), 5465-5467.

Mise à jour le 21 janvier 2014