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Accueil du site > Publications > 2- Criblages de chimiothèques > 2009

Publications 2009

1. Keriel, F. Mahuteau-Betzer, C. Jacquet, M. Plays, D. Grierson, M. Sitbon, J. Tazi
Protection against Retrovirus Pathogenesis by SR Protein Inhibitors
PLoS One 2009, 2, 4, e4533.

2. T.M. HOANG, B. FAVIER, A. VALETTE, C. BARETTE, C.H. NGUYEN, L. LAFANECHERE, D.S. GRIERSON, S. DIMITROV , A. MOLLA
Benzo [e]pyridoindoles, novel inhibitors of the aurora kinases
Cell Cycle 2009, 8 (5), 765-772.

3. Cohen, Anita ; Crozet, Maxime D. ; Rathelot, Pascal ; Vanelle, Patrice
An efficient aqueous microwave-assisted Suzuki-Miyaura cross-coupling reaction in the thiazole series
Green Chemistry 2009, 11(11), 1736-1742.

4. Crozet, Maxime D. ; Zink, Laura ; Remusat, Vincent ; Curti, Christophe ; Vanelle, Patrice
Efficient microwave-assisted palladium-catalyzed Suzuki-Miyaura cross-coupling reactions in 5-nitroimidazole series
Synthesis 2009,18, 3150-3156.

5. Khoumeri, Omar ; Crozet, Maxime D. ; Terme, Thierry ; Vanelle, Patrice _ Original TDAE application : synthesis of 2-substituted-4,11-dimethoxy-anthra[2,3-b]furan-5,10-diones via intramolecular Buchwald reaction _ Tetrahedron Letters 2009,50(46), 6372-6376.

6. Kabri, Youssef ; Gellis, Armand ; Vanelle, Patrice
Synthesis of Original 2-Substituted 4-Arylquinazolines by Microwave-Irradiated Suzuki-Miyaura Cross-Coupling Reactions
European Journal of Organic Chemistry 2009, 24, 4059-4066.

7. Since, Marc ; Terme, Thierry ; Vanelle, Patrice
Original TDAE strategy using α-halocarbonyl derivatives
Tetrahedron 2009, 65(31), 6128-6134.

8. Juspin, Thierry ; Terme, Thierry ; Vanelle, Patrice
TDAE strategy using α-diketones : rapid access to 2,3-diphenyl quinoline and acenaphtho[1,2-b]quinoline derivatives
Synlett 2009,9, 1485-1489.

9. Verhaeghe, Pierre ; Azas, Nadine ; Hutter, Sebastien ; Castera-Ducros, Caroline ; Laget, Michele ; Dumetre, Aurelien ; Gasquet, Monique ; Reboul, Jean-Pierre ; Rault, Sylvain ; Rathelot, Pascal ; et al
Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines
Bioorganic & Medicinal Chemistry 2009, 17(13), 4313-4322.

10. C. Rochais, D.-N. Vu, E. Lescot, J. Sopkova de Oliveira Santos, R. Bureau, L. Meijer, P. Dallemagne, S. Rault
Synthesis of New DiPyrrolo- and FuroPyrroloPyrazinones Related to Tripentones and their Biological Evaluation as Potential (CDKs1–5, GSK-3) Kinases Inhibitors
European Journal of Medicinal Chemistry, 2009, 44, 708-716.

11. S. Lemaitre, A. Lepailleur, R. Bureau, S. Butt-Gueulle, V. Lelong-Boulouard, P. Duchatelle, M. Boulouard, A. Dumuis, C. Daveu, F. Lezoualc’h, B. Pfeiffer, F. Dauphin, S. Rault
Novel antagonists of serotonin-4 receptors : Synthesis and biological evaluation of pyrrolothienopyrazines
Bioorganic and Medicinal Chemistry, 2009, 17(6), 2607-2622.

12. C. Rochais, P. Dallemagne, S. Rault.
Tripentones : A Promising Series of Potent Anti-Cancer Agents
Anti-Cancer Agents in Medicinal Chemistry, 2009, 9, 369-380.

13. V. Perri, C. Rochais, T. Cresteil, P. Dallemagne, S. Rault
Synthesis, reactivity and biological evaluation of novel halogenated tripentones
Bioorganic and Medicinal Chemistry, 2009, 17, 7783–7788.

Mise à jour le 1er juillet 2014