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Accueil du site > Publications > 2- Criblages de chimiothèques > 2008

Publications 2008

1. R. PRUDENT, V. MOUCADEL, M. LOPEZ RAMOS, S. ACI, B. LAUDET, L. MOUAWAD, C. BARETTE, J. EINHORN, C. EINHORN, J.-N. DENIS, G. BISSON, F. SCHMIDT, S. ROY, L. LAFANECHERE, J.-C. FLORENT, C. COCHET
Expanding the chemical diversity of CK2 inhibitors
Mol Cell Biochem 2008, 316, 71-85.

2. R. PRUDENT, M. LOPEZ-RAMOS, V. MOUCADEL, C. BARETTE, D. GRIERSON, L. MOUAWAD, J.-C. FLORENT, L. LAFANECHERE, F. SCHMIDT, C. COCHET
Salicylaldehyde Derivatives as New Protein Kinase CK2 Inhibitors
Biochim. Biophys Acta 2008, 1780, 1412-1420.

3. P. Verhaerghe, N. Azas, M. Gasquet, S. Hutter, C. Ducros, M. Laget, S. Rault, P. Rathelot, P. Vanelle
Synthesis and antiplasmodial activity of new 4-aryl-2-trichlorométhyl quinazolines
Bioorganic and Medicinal Chemistry Letters, 2008, 18, 396-401.

4. E. Lescot, R. Bureau, S. Rault
Nonpeptide Urotensin-II receptor agonists and antagonists : Rewiew and structure-activity relationships
Peptides, 2008, 29, 680-690.

5. R. Bureau, T. Varin, A. Lepailleur, C. Daveu, S. Lemaitre, J.-C. Lancelot, A. Lesnard, S. Butt-Gueulle, F. Dauphin, S. Rault
Pharmacophores of 5HT4 ligands : Experience of CERMN and implications for drug design
Current Computer-Aided Drug Design, 2008, 4, 199-208.

6. E. Lescot, J. Sopkova-de Oliveira Santos, N. Colloc’h, J. Rodrigo, I. Milazzo-Segalas, R. Bureau, S. Rault
Three-dimensional model of human urotensin-II receptor : Docking of human urotensin-II and nonpeptide antagonists in the binding site and comparison with an antagonist pharmacophore model
Proteins : Structure, Function, and Bioinformatics, 2008, 73(1), 173-184.

7. T. Varin, N. Saettel, J. Villain, A. Lesnard, F. Dauphin, R. Bureau, S. Rault
3D Pharmacophore, hierarchical methods, and 5-HT4 receptor binding data
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 23(5), 593-603.

8. L. El Kihel, M. Clément, M.-A. Bazin, G. Descamps, M. Khalid, S. Rault
New lithocholic and chenodeoxycholic piperazinylcarboxamides with antiproliferative and pro-apoptotic effects on human cancer cell lines
Bioorganic and Medicinal Chemistry, 2008, 16(18), 8737-8744.

9. Z. Omran, S. Stiebing, A.-M. Godard, J. Sopkova-de Oliveira Santos, P. Dallemagne
Synthesis and biological evaluation of new Donepezil-like Thiaindanones as AChE inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 23(5), 696-703.

Mise à jour le 21 janvier 2015